P-gp modulator 2 (Compound 27) is a potent, competitive, allostericP-glycoprotein(P-gp)modulator^[1].

P-gp modulator 2 (Compound 27) shows cytotoxicity on L5178Y parental (L5178Y-PAR) and human ABCB1-gene transfected (L5178Y-MDR) mouse T-lymphoma cells with IC₅₀values of 8.0 ± 1.1 and 10.7 ± 1.1 μM, respectively^[1].

470.32

C₂₂H₂₀BrN₃O₄

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.