S1427 is a tranylcypromine-derivedLSD1inhibitor with theIC₅₀of 390 nM andK_iof 80 nM. S1427 exhibits desirable hERG channel inhibition and microsomal stability profiles. Inhibition of LSD1 partially reduces the proliferation ofcancercells^[1].

474.52

C₂₅H₂₉F₃N₄O₂

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.