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GABAA receptor agent 1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GABAA receptor agent 1图片
CAS NO:1571-87-5
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议

产品介绍
GABAAreceptoragent1是GABAA受体的高亲和力配体,具有较强的抗惊厥活性。
Cas No.1571-87-5
别名2-(4-氯苯基)-6-硝基-1H-苯并[D]咪唑
Canonical SMILESO=[N+](C1=CC=C2N=C(C3=CC=C(Cl)C=C3)NC2=C1)[O-]
分子式C13H8ClN3O2
分子量273.67
溶解度DMSO: 83.33 mg/mL (304.49 mM)
储存条件Store at -20℃
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述

GABAA receptor agent 1 is a high affinity ligand for GABAA receptor, with potent anticonvulsant activity[1].

GABAA receptor agent 1 (30 mg/kg; intraperitoneal) inhibits the maximum electroshock (MES) and pentylenetetrazole (PTZ)-induced convulsions in swiss albino rats[1].

[1]. Jain P, et al. Design, synthesis and biological evaluation of some novel benzimidazole derivatives for their potential anticonvulsant activity. Arch Pharm Res. 2010 Jul;33(7):971-80.