Volinanserin-d4 (MDL100907-d4) hydrochloride is the deuterium labeled Volinanserin hydrochlorid. Volinanserin is a potent and selective antagonist of5-HT₂receptor, with aK_iof 0.36 nM, and shows 300-fold selectivity for5-HT₂receptorover 5-HT_1c, alpha-1 and DA D₂receptors. Volinanserin has antipsychotic activity^[1][2].

Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs^[1].

413.95

C₂₂H₂₅D₄ClFNO₃

1217617-73-6

氟利色林 d4 (盐酸盐)

Room temperature in continental US; may vary elsewhere.

Please store the product under the recommended conditions in the Certificate of Analysis.